Enzymology in drug discovery [electronic resource] : part 2 of 2 / Robert A. Copeland.
Material type:![Film](/opac-tmpl/lib/famfamfam/VM.png)
- Enzymology in drug discovery part, part 2 of 2
- Drugs -- Design
- Enzyme inhibitors -- Structure-activity relationships
- Enzyme inhibitors -- Therapeutic use
- Enzymes
- Enzymology
- Pharmaceutical chemistry
- Drug Design
- Drug Discovery
- Enzyme Inhibitors -- chemistry
- Enzyme Inhibitors -- metabolism
- Enzyme Inhibitors -- pharmacology
- Enzyme Inhibitors -- therapeutic use
Animated audio-visual presentation with synchronized narration.
Title from title frames.
Contents: Enzymes as targets for drug discovery -- Protein-ligand binding equilibria -- Enzyme reaction mechanisms -- Structure and function of enzyme active sites -- Measuring enzyme velocity in the laboratory -- Reversible modes of enzyme inhibition -- Enzyme inhibition as a mechanism of pharmacological intervention in disease -- Clinical value of different inhibition modalities -- Non-classical inhibition -- Enzyme assays and screening criteria -- Lead optimization -- Summary: basic information to look for.
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Mode of access: World Wide Web.
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